SCHEMBL6441973

SCHEMBL6441973

CS(=O)(=O)C(CNC(=O)c1ccccc1[N+](=O)[O-])C(=O)NCC#N

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.48
ALDH1A1 P00352 5/20 0.47
LMNA P02545 4/20 0.47
HPGD P15428 3/20 0.46
HTT P42858 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
CTSB P07858 1/20 0.43
MAPT P10636 2/20 0.43
GAA P10253 2/20 0.43
SLC12A2 P55011 1/20 0.43
SLC12A5 Q9H2X9 1/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444783 0.90 ALDH1A1 (0.47) CTSDALDH1A1LMNAHPGDHTT
SCHEMBL6446549 0.84 KDM4E (0.50) HTTMEN1KMT2ACTSBKDM4E
SCHEMBL6445609 0.83 CTSK (0.52) CTSDALDH1A1LMNAHPGDHTT
SCHEMBL6447040 0.83 CTSD (0.49) CTSDALDH1A1LMNAHPGDHTT
SCHEMBL6442213 0.82 NPC1 (0.45) LMNAHPGDCTSBGAAKDM4E
SCHEMBL6020500 0.81 CTSS (0.52) CTSDALDH1A1CTSB
SCHEMBL6442065 0.80 CTSL (0.54) CTSB
SCHEMBL6445280 0.79 CTSK (0.51) CTSDALDH1A1LMNAHPGDHTT
SCHEMBL6737541 0.78 CTSL (0.43) ALDH1A1HPGDCTSB
SCHEMBL6441987 0.77 CTSK (0.46) CTSDALDH1A1LMNAHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed