SCHEMBL6463841

SCHEMBL6463841

CCCCN(C(=O)O)C(=O)N[C@@H](CCc1ccccc1)C(O)c1nc(C(=O)NC(c2ccccc2)c2ccccc2)co1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 6/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HPGDS O60760 1/20 0.33
MMP2 P08253 2/20 0.33
MMP3 P08254 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KMT2A Q03164 1/20 0.32
LONP1 P36776 1/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ASAH1 Q13510 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6463773 0.83 DAGLA (0.34) CYP1A2CYP2C9CYP2C19KMT2ALONP1
SCHEMBL6465469 0.82 PPARG (0.35) CYP1A2CYP2C9CYP2C19KMT2ALONP1
SCHEMBL6465287 0.81 TRPV1 (0.42) LONP1
SCHEMBL6463837 0.71 NPSR1 (0.35) C3AR1HDAC1HDAC8HDAC6HPGDS
SCHEMBL7046400 0.70 PTGER4 (0.38) HDAC1HDAC8HDAC6NPSR1
SCHEMBL6467305 0.70 MMP9 (0.44) C3AR1HDAC1HDAC8HDAC6MMP2
SCHEMBL6467310 0.70 MMP9 (0.44) C3AR1HDAC1HDAC8HDAC6MMP2
SCHEMBL6466256 0.70 MMP9 (0.44) C3AR1HDAC1HDAC8HDAC6MMP2
SCHEMBL7466136 0.69 FAAH (0.36) CYP3A4
SCHEMBL6466197 0.69 FAAH (0.36) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed