SCHEMBL6465103

SCHEMBL6465103

CCCC[C@H](C(=O)c1nc2ccccc2o1)C(CS(=O)(=O)Cc1ccccc1)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.41
CES1 P23141 2/20 0.41
DAGLA Q9Y4D2 1/20 0.41
XDH P47989 3/20 0.40
ALDH1A1 P00352 1/20 0.40
CTSS P25774 10/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690593 0.78 FAAH (0.38) FAAHCES1DAGLAXDHALDH1A1
SCHEMBL6467110 0.76 CTSS (0.44) FAAHCES1CTSSCYP3A4CYP2C9
SCHEMBL6465112 0.76 CTSS (0.47) FAAHCES1DAGLAALDH1A1CTSS
SCHEMBL5413826 0.76 CTSS (0.46) CTSSCYP3A4CYP2C9
SCHEMBL7187229 0.75 CTSS (0.43) FAAHCES1DAGLACTSSCYP3A4
SCHEMBL6466904 0.74 DAGLA (0.50) FAAHCES1DAGLAXDH
SCHEMBL6465885 0.74 XDH (0.47) FAAHCES1DAGLAXDHCTSS
SCHEMBL6463186 0.74 CTSS (0.50) CTSSCYP3A4CYP2C9
SCHEMBL6467933 0.73 CTSS (0.44) CTSSCYP3A4CYP2C9
SCHEMBL6691866 0.73 CTSS (0.44) CTSSCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed