SCHEMBL6465121

SCHEMBL6465121

CC[C@H](NC(=O)N(CCS(=O)(=O)Cc1c(C)noc1C)C(=O)O)C(=O)c1nc2ccccc2o1

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSS P25774 20/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045892 0.92 CTSS (0.41) CTSSCYP3A4CYP2C9
SCHEMBL6465108 0.82 XDH (0.39)
SCHEMBL6468436 0.80 CTSS (0.44) CTSSCYP3A4CYP2C9
SCHEMBL7116648 0.79 CTSS (0.43) CTSSCYP3A4CYP2C9
SCHEMBL7116654 0.79 CTSS (0.43) CTSSCYP3A4CYP2C9
SCHEMBL6464424 0.78 CTSS (0.43) CTSSCYP3A4CYP2C9
SCHEMBL6464410 0.78 FAAH (0.42) CTSSCYP3A4CYP2C9
SCHEMBL6462828 0.76 CTSS (0.41) CTSSCYP3A4CYP2C9
SCHEMBL6462867 0.74 CTSS (0.41) CTSSCYP3A4CYP2C9
SCHEMBL7046208 0.74 CTSS (0.38) CTSSCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed