SCHEMBL6465108

SCHEMBL6465108

CCCN(C(=O)c1nc2ccccc2o1)C(=O)N(CCS(=O)(=O)Cc1c(C)noc1C)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.39
AR P10275 1/20 0.36
HSF1 Q00613 5/20 0.34
FAAH O00519 2/20 0.34
CES1 P23141 1/20 0.34
ALDH1A1 P00352 3/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
TAS2R8 Q9NYW2 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6465121 0.82 CTSS (0.45)
SCHEMBL6465186 0.81 ALDH1A1 (0.44) XDHHSF1FAAHCES1ALDH1A1
SCHEMBL7045889 0.78 NPC1 (0.34) XDHARHSF1FAAHCES1
SCHEMBL14110445 0.78 FAAH (0.47) XDHHSF1FAAHCES1ALDH1A1
SCHEMBL6464421 0.77 ALDH1A1 (0.44) XDHFAAHCES1ALDH1A1GAA
SCHEMBL6464404 0.77 DAGLA (0.48) XDHFAAHCES1ALDH1A1
SCHEMBL6462825 0.76 XDH (0.38) XDHHSF1FAAHCES1ALDH1A1
SCHEMBL7045892 0.76 CTSS (0.41)
SCHEMBL6466172 0.73 FAAH (0.36) XDHHSF1FAAHCES1ALDH1A1
SCHEMBL14110504 0.71 FAAH (0.51) XDHHSF1FAAHCES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed