SCHEMBL6472183

SCHEMBL6472183

O=C(CCC1CCCCC1)N[C@@H](CCc1ccccc1)C(=O)c1ncco1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 12/20 0.48
CES1 P23141 2/20 0.45
NCEH1 Q6PIU2 1/20 0.45
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
HPGD P15428 1/20 0.43
CTSL P07711 2/20 0.42
CTSB P07858 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
EPHX2 P34913 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048644 0.83 FAAH (0.47) FAAHCES1MEN1KMT2ACTSL
SCHEMBL6462775 0.83 CES1 (0.47) CES1MEN1KMT2ACTSLCTSB
SCHEMBL7044248 0.82 CTSL (0.49) CTSLCTSBCTSS
SCHEMBL6468629 0.81 CTSS (0.48) FAAHCES1MEN1KMT2ACTSL
SCHEMBL6465141 0.81 CTSS (0.48) FAAHCES1MEN1KMT2ACTSL
SCHEMBL6463419 0.81 CTSS (0.48) FAAHCES1MEN1KMT2ACTSL
SCHEMBL7045305 0.80 DAGLA (0.52) CES1MEN1KMT2AHPGDCTSL
SCHEMBL6462673 0.80 MEN1 (0.42) FAAHMEN1KMT2AHPGDCTSL
SCHEMBL6464884 0.80 CTSS (0.49) FAAHCES1MEN1KMT2ACTSL
SCHEMBL7045308 0.78 CTSS (0.49) MEN1KMT2ACTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed