SCHEMBL6462775

SCHEMBL6462775

O=C(CCC1CCCCC1)NC(CCc1ccccc1)C(=O)c1nc(C(=O)O)co1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.47
EPHX2 P34913 1/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
DAGLA Q9Y4D2 4/20 0.40
CTSL P07711 3/20 0.40
CTSB P07858 3/20 0.40
CTSS P25774 3/20 0.40
CTSK P43235 3/20 0.40
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RAB9A P51151 1/20 0.38
MMP2 P08253 2/20 0.38
BMP1 P13497 1/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
TBXA2R P21731 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045305 0.91 DAGLA (0.52) CES1EPHX2ALDH1A1MEN1KMT2A
SCHEMBL6472183 0.83 FAAH (0.48) CES1EPHX2ALDH1A1MEN1KMT2A
SCHEMBL6465141 0.81 CTSS (0.48) CES1EPHX2MEN1KMT2ADAGLA
SCHEMBL6468629 0.81 CTSS (0.48) CES1EPHX2MEN1KMT2ADAGLA
SCHEMBL6463419 0.81 CTSS (0.48) CES1EPHX2MEN1KMT2ADAGLA
SCHEMBL6473243 0.81 BMP1 (0.41) CES1EPHX2ALDH1A1MEN1KMT2A
SCHEMBL6464884 0.80 CTSS (0.49) CES1MEN1KMT2ADAGLACTSL
SCHEMBL6464300 0.80 CTSS (0.44) MEN1KMT2ADAGLACTSLCTSB
SCHEMBL7048644 0.80 FAAH (0.47) CES1ALDH1A1MEN1KMT2ATDP1
SCHEMBL7045308 0.78 CTSS (0.49) MEN1KMT2ADAGLACTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed