SCHEMBL6477967

SCHEMBL6477967

CC(C)CC(NC(=O)O)C(=O)NC(CCc1ccccc1)C(=O)c1nc(C(=O)NCCCc2ccccc2)co1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 7/20 0.44
CTSL P07711 2/20 0.43
CTSB P07858 2/20 0.43
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
MMP2 P08253 2/20 0.43
MMP8 P22894 2/20 0.42
CES1 P23141 1/20 0.42
ANPEP P15144 1/20 0.42
DAGLA Q9Y4D2 2/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464784 0.95 ANPEP (0.48) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6063167 0.90 CTSL (0.51) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6466269 0.88 MMP9 (0.44) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6464783 0.88 MMP9 (0.44) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6466271 0.88 MMP9 (0.44) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6063868 0.85 PSMB5 (0.44) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6061873 0.85 CA5A (0.53) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6064394 0.85 CA5A (0.53) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6463220 0.82 CTSL (0.51) MMP3CTSLCTSBCTSSCTSK
SCHEMBL6464780 0.81 CTSB (0.42) MMP3CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed