SCHEMBL6485457

SCHEMBL6485457

CC(C)(C)N(Cc1cccc(NC(=O)C(=O)Nc2ccc(-c3cnco3)cc2)c1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 15/20 0.56
IMPDH1 P20839 10/20 0.56
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
PKM P14618 1/20 0.47
PORCN Q9H237 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
AAK1 Q2M2I8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6484655 0.91 IMPDH2 (0.64) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL6485360 0.86 IMPDH2 (0.68) IMPDH2IMPDH1AAK1
SCHEMBL6493937 0.83 IMPDH2 (0.52) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL6494993 0.83 IMPDH2 (0.56) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL6499362 0.80 IMPDH2 (0.59) IMPDH2IMPDH1NPC1RAB9AKDM4E
Trifluoroacetic Acid SCHEMBL27561206 0.78 IMPDH2 (0.53) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL27542606 0.78 IMPDH2 (0.64) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL6486557 0.76 IMPDH2 (0.54) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL6497151 0.73 IMPDH2 (1.00) IMPDH2IMPDH1NPC1RAB9AKDM4E
SCHEMBL6500618 0.73 IMPDH2 (0.72) IMPDH2IMPDH1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6867299-B2 Inosine monophosphate dehydrogenase (IMPDH); use as immunosuppressants, anticancer agents and antiviral agents HOFFMANN-LA ROCHE INC. (US) 2005-03-15 US disclosed