SCHEMBL6496283

SCHEMBL6496283

CN1CN(Cc2ccccc2)CC2=C1CCN(C(=O)OCc1ccc(OC(F)(F)F)cc1)C2

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.45
PTGDR2 Q9Y5Y4 5/20 0.43
ENPP2 Q13822 1/20 0.42
ATXN2 Q99700 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TMEM97 Q5BJF2 5/20 0.41
SIGMAR1 Q99720 5/20 0.41
TNF P01375 1/20 0.41
NOD2 Q9HC29 1/20 0.41
NOD1 Q9Y239 1/20 0.41
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
P2RY1 P47900 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
BACE1 P56817 1/20 0.40
LSS P48449 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6496169 0.90 TMEM97 (0.48) ALDH1A1TMEM97SIGMAR1
SCHEMBL6489104 0.89 SIGMAR1 (0.46) PTGDR2TMEM97SIGMAR1TSHR
SCHEMBL6496625 0.87 TMEM97 (0.45) PTGDR2TMEM97SIGMAR1
SCHEMBL6487154 0.85 TMEM97 (0.43) PTGDR2ALDH1A1TMEM97SIGMAR1
SCHEMBL6495760 0.84 TMEM97 (0.44) TMEM97SIGMAR1
SCHEMBL6487210 0.83 PTGDR2 (0.42) CHRM4PTGDR2ENPP2ATXN2TMEM97
SCHEMBL6487473 0.82 SIGMAR1 (0.47) PTGDR2ALDH1A1TMEM97SIGMAR1
SCHEMBL6488679 0.82 TMEM97 (0.39) PTGDR2ALDH1A1TMEM97SIGMAR1TSHR
SCHEMBL6490718 0.80 ALDH1A1 (0.39) ALDH1A1TMEM97SIGMAR1TSHR
SCHEMBL6502757 0.79 TMEM97 (0.39) ALDH1A1TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6869958-B2 Fused tetrahydropyridine derivatives as matrix metalloproteinase inhibitors WARNER-LAMBERT COMPANY (US) 2005-03-22 US disclosed
US-20040038960-A1 Fused tetrahydropyridine derivatives as matrix metalloproteinase inhibitors LI JIE JACK (US) 2004-02-26 US disclosed
WO-2004014909-A1 FUSED TETRAHYDROPYRIDINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040038960-A1 Fused tetrahydropyridine derivatives as matrix metalloproteinase inhibitors MMP9, MMP3, MMP13 CHRM4 2157/4885PTGDR2 591/4885ENPP2 974/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.