SCHEMBL6497472

SCHEMBL6497472

[CH2]NC(=O)c1ccc(SC(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.56
KCNK2 O95069 12/20 0.55
KCNK10 P57789 9/20 0.55
EPHX2 P34913 1/20 0.52
NR1H4 Q96RI1 1/20 0.52
KIF11 P52732 1/20 0.46
PTPRZ1 P23471 2/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PTPN1 P18031 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13485813 0.83 TRPV1 (0.58) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL21995806 0.81 TRPV1 (0.56) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL6497474 0.81 PLK1 (0.61) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL10919991 0.78 LMNA (0.53) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL1015553 0.76 KCNK2 (0.57) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL10740573 0.76 ALDH1A1 (0.50) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL6495770 0.76 CES2 (0.61) TRPV1EPHX2NPC1RAB9APTPN1
SCHEMBL16610094 0.76 EPHX2 (0.58) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL16341732 0.75 TRPV1 (0.57) TRPV1KCNK2KCNK10EPHX2NR1H4
SCHEMBL2541283 0.75 KIF11 (0.54) TRPV1KCNK2KCNK10EPHX2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed