SCHEMBL6504314

SCHEMBL6504314

O=C(O)[C@H](Cc1ccc2oc(CCCNc3nc4ccccc4[nH]3)cc(=O)c2c1)NS(=O)(=O)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.44
ITGAV P06756 11/20 0.44
ITGB1 P05556 1/20 0.41
ITGA5 P08648 1/20 0.41
ITGA2B P08514 2/20 0.37
PIN1 Q13526 1/20 0.37
KCNH2 Q12809 1/20 0.36
TEAD4 Q15561 1/20 0.35
BCHE P06276 1/20 0.35
TRPC3 Q13507 1/20 0.35
TRPC4 Q9UBN4 1/20 0.35
TRPC5 Q9UL62 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6503005 0.91 ITGB3 (0.51) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL6505393 0.91 ITGB3 (0.42) ITGB3ITGAVITGB1ITGA5KCNH2
SCHEMBL6495002 0.91 ITGB3 (0.41) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL6506524 0.87 ITGB3 (0.40) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL5204669 0.83 ITGB1 (0.49) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL3048231 0.82 ITGB3 (0.45) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL6505728 0.78 ITGB3 (0.49) ITGB3ITGAVITGA2B
SCHEMBL14431792 0.78 BCHE (0.37) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL5204539 0.77 ITGB3 (0.41) ITGB3ITGAVITGB1ITGA5ITGA2B
SCHEMBL6495597 0.76 ITGB3 (0.39) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849646-B1 Chromenone and chromanone derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2005-02-01 US disclosed
EP-1124824-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2001-08-22 EP disclosed
WO-2000026212-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2000-05-11 WO disclosed