SCHEMBL6495002

SCHEMBL6495002

CCCCS(=O)(=O)N[C@@H](Cc1ccc2oc(CCCNc3nc4ccccc4[nH]3)cc(=O)c2c1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.41
ITGAV P06756 12/20 0.41
BCHE P06276 1/20 0.41
TRPC3 Q13507 1/20 0.41
TRPC4 Q9UBN4 1/20 0.41
TRPC5 Q9UL62 1/20 0.41
ITGA2B P08514 6/20 0.39
ITGB1 P05556 2/20 0.38
ITGA5 P08648 2/20 0.38
CHRM2 P08172 1/20 0.35
SLC6A4 P31645 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504314 0.91 ITGB3 (0.44) ITGB3ITGAVBCHETRPC3TRPC4
SCHEMBL6505393 0.90 ITGB3 (0.42) ITGB3ITGAVBCHETRPC3TRPC4
SCHEMBL6503005 0.89 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL3039366 0.86 ITGB3 (0.40) ITGB3ITGAVITGA2BCHRM2SLC6A4
SCHEMBL5204428 0.83 ITGB1 (0.47) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL3048231 0.81 ITGB3 (0.45) ITGB3ITGAVBCHEITGA2BITGB1
SCHEMBL7542370 0.78 BCHE (0.43) ITGB3ITGAVBCHETRPC3TRPC4
SCHEMBL6506524 0.78 ITGB3 (0.40) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL5204539 0.78 ITGB3 (0.41) ITGB3ITGAVBCHETRPC3TRPC4
SCHEMBL14431792 0.77 BCHE (0.37) ITGB3ITGAVBCHETRPC3TRPC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849646-B1 Chromenone and chromanone derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2005-02-01 US disclosed
EP-1124824-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2001-08-22 EP disclosed
WO-2000026212-A1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2000-05-11 WO disclosed