SCHEMBL650647

SCHEMBL650647

O=S(=O)(Cl)c1ncccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 19/20 0.47
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28502273 0.83 NFE2L2 (0.43) NFE2L2LMNA
SCHEMBL6098339 0.81 LMNA (0.50) NFE2L2LMNA
SCHEMBL950477 0.81 NFE2L2 (0.45) NFE2L2LMNA
Hydrochloric Acid SCHEMBL7085595 0.81 NFE2L2 (0.42) NFE2L2LMNA
SCHEMBL30727252 0.78 NFE2L2 (0.44) NFE2L2LMNA
SCHEMBL27327034 0.78 NFE2L2 (0.44) NFE2L2LMNA
SCHEMBL1039344 0.77 NOS3 (0.43) NFE2L2
SCHEMBL9734435 0.77 TRPV4 (0.42) NFE2L2
SCHEMBL30665364 0.77 TRPV4 (0.42) NFE2L2LMNA
SCHEMBL937654 0.77 TRPV4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1048654-B1 Process for the preparation of chloropyridine sulfonyl chloride RUETGERS ORGANICS GMBH (DE) 2003-07-30 EP claimed
US-6310214-B1 FROM HYDROXYPYRIDINESULPHONIC ACIDS COMPRISING PASSING CHLORINE GAS INTO A MIXTURE OF A HYDROXYPYRIDINESULPHONIC ACID AND OF PHOSPHORUS TRICHLORIDE; HEATING; DISTILLATION RUETGERS ORGANICS GMBH (DE) 2001-10-30 US claimed
EP-1048654-A2 Process for the preparation of chloropyridine sulfonyl chloride Rütgers Organics GmbH (DE) 2000-11-02 EP claimed
WO-2000063177-A1 METHOD OF PRODUCING CHLOROPYRIDINE SULFONIC ACID CHLORIDES RÜTGERS ORGANICS GMBH (DE) 2000-10-26 WO claimed
US-9174964-B2 AMPK-activating piperidinyloxy-substituted 2,3-dihydro-1H-indene-1-amine compounds and pharmaceutical compositions including the same RIGEL PHARMACEUTICALS, INC. (US) 2015-11-03 US disclosed
US-20150252019-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CELGENE AVILOMICS RESEARCH, INC. 2015-09-10 US disclosed
EP-2231600-B1 CARBOXAMIDE, SULFONAMIDE AND AMINE COMPOUNDS FOR METABOLIC DISORDERS RIGEL PHARMACEUTICALS INC (US) 2015-07-29 EP disclosed
US-9067929-B2 Heterocyclic compounds and uses thereof CELGENE AVILOMICS RESEARCH, INC. (US) 2015-06-30 US disclosed
CN-101039904-B Is suitable for treating dopamine D3Heterocyclic compounds for receptor-modulated responsive disorders ABBOTT GMBH & CO KG 2014-09-24 CN disclosed
US-20140073661-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CELGENE AVILOMICS RESEARCH, INC. (US) 2014-03-13 US disclosed
US-20140051673-A1 AMPK-Activating Heterocycloalkyloxy(Hetero)Aryl Carboxamide, Sulfonamide And Amine Compounds And Methods For Using The Same RIGEL PHARMACEUTICALS, INC. (US) 2014-02-20 US disclosed
US-8586600-B2 Heterocyclic compounds and uses thereof CELGENE AVILOMICS RESEARCH, INC. (US) 2013-11-19 US disclosed
US-6310214-B1 FROM HYDROXYPYRIDINESULPHONIC ACIDS COMPRISING PASSING CHLORINE GAS INTO A MIXTURE OF A HYDROXYPYRIDINESULPHONIC ACID AND OF PHOSPHORUS TRICHLORIDE; HEATING; DISTILLATION RUETGERS ORGANICS GMBH (DE) 2001-10-30 US disclosed
US-6310214-B1 FROM HYDROXYPYRIDINESULPHONIC ACIDS COMPRISING PASSING CHLORINE GAS INTO A MIXTURE OF A HYDROXYPYRIDINESULPHONIC ACID AND OF PHOSPHORUS TRICHLORIDE; HEATING; DISTILLATION RUETGERS ORGANICS GMBH (DE) 2001-10-30 US disclosed
WO-2000063177-A8 METHOD OF PRODUCING CHLOROPYRIDINE SULFONIC ACID CHLORIDES RUETGERS ORGANICS GMBH (DE) 2001-02-22 WO disclosed
EP-1048654-A3 Process for the preparation of chloropyridine sulfonyl chloride Rütgers Organics GmbH (DE) 2000-11-08 EP disclosed
EP-1048654-A2 Process for the preparation of chloropyridine sulfonyl chloride Rütgers Organics GmbH (DE) 2000-11-02 EP disclosed
WO-2000063177-A1 METHOD OF PRODUCING CHLOROPYRIDINE SULFONIC ACID CHLORIDES RÜTGERS ORGANICS GMBH (DE) 2000-10-26 WO disclosed
WO-1997046553-A1 THROMBIN INHIBITORS NOVARTIS AG (CH) 1997-12-11 WO disclosed
US-4490380-A 3-CHLORO-2-PYRIDINE SULFONAMIDE; MITICIDES; LARVACIDES THE DOW CHEMICAL COMPANY (US) 1984-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150252019-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ABCG2, CYP3A5, CYP3A43 NFE2L2 2429/4885LMNA 1530/4885
US-20140051673-A1 AMPK-Activating Heterocycloalkyloxy(Hetero)Aryl Carboxamide, Sulfonamide And Amine Compounds And Methods For Using The Same PRKAA1, PRKAA2, PRKAG1 NFE2L2 687/4885LMNA 2643/4885
US-20140073661-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ABCG2, CYP3A5, CYP3A43 NFE2L2 2429/4885LMNA 1530/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.