SCHEMBL6507499

SCHEMBL6507499

CC(COc1ccccc1)O[Si](C)(C)C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.49
CYP2D6 P10635 4/20 0.46
MAOA P21397 1/20 0.45
PTGS1 P23219 1/20 0.45
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
SCN4A P35499 2/20 0.40
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
NPC1 O15118 1/20 0.36
MTOR P42345 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC22A2 O15244 1/20 0.36
SLC22A1 O15245 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22249309 0.84 KDM4E (0.36) LMNACYP2D6CYP2C9CYP2C19NPC1
SCHEMBL22233284 0.84 ALDH1A1 (0.43) LMNAMAPK1ALDH1A1SMN1; SMN2TSHR
SCHEMBL6490888 0.83 CYP2D6 (0.43) LMNACYP2D6MAOAPTGS1MTNR1A
SCHEMBL22233863 0.80 CA2 (0.39) LMNACYP2D6CYP2C9CYP2C19NPC1
SCHEMBL3603475 0.80 ALDH1A3 (0.42) LMNACYP2D6ADRB2ADRB1ADRB3
SCHEMBL1931571 0.80 ALDH1A3 (0.42) LMNACYP2D6ADRB2ADRB1ADRB3
SCHEMBL19750656 0.80 LMNA (0.44) LMNAHSD17B10ALDH1A1
SCHEMBL817869 0.80 CYP2D6 (0.43) LMNACYP2D6MAOAPTGS1MTNR1A
SCHEMBL714416 0.80 CYP2D6 (0.43) LMNACYP2D6MAOAPTGS1MTNR1A
SCHEMBL8429746 0.80 CYP2D6 (0.43) LMNACYP2D6MAOAPTGS1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016885-A2 COMPOUNDS WITH COMBINED CALCIUM CHANNEL BLOCKER AND β-ADRENERGIC ANTAGONIST OR PARTIAL AGONIST ACTIVITIES FOR TREATMENT OF HEART DISEASE ARTESIAN THERAPEUTICS, INC. (US) 2005-02-24 WO disclosed