SCHEMBL6508617

SCHEMBL6508617

COc1cc(OC)nc(NC(N)=Nc2cccc(Cc3ccccc3)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.46
GRIN2D O15399 3/20 0.46
GRIN3B O60391 3/20 0.46
GRIN1 Q05586 3/20 0.46
GRIN2A Q12879 3/20 0.46
GRIN2B Q13224 3/20 0.46
GRIN2C Q14957 3/20 0.46
GRIN3A Q8TCU5 3/20 0.46
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
HTT P42858 1/20 0.41
NOS1 P29475 3/20 0.41
KMT2A Q03164 1/20 0.40
CYP1A2 P05177 1/20 0.39
NOS2 P35228 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510588 0.84 LMNA (0.50) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6507347 0.80 LMNA (0.52) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6513739 0.76 SMN1; SMN2 (0.42) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6515320 0.74 SIGMAR1 (0.46) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6507406 0.74 RAB9A (0.52) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL5923340 0.74 MAPT (0.44) MAPTTP53GLAHTTKMT2A
SCHEMBL6507964 0.73 SIGMAR1 (0.72) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9392429 0.72 SIGMAR1 (0.56) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL14861786 0.72 SIGMAR1 (0.65) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9392449 0.70 SIGMAR1 (0.50) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095345-A2 HETEROARYL GUANIDINES AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS, INC. (US) 2005-10-13 WO claimed