SCHEMBL6522978

SCHEMBL6522978

O=C(O)CCC1=CSc2ccccc2-c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
PTGER1 P34995 4/20 0.42
PTGER4 P35408 4/20 0.42
PTGER3 P43115 4/20 0.42
PTGER2 P43116 4/20 0.42
FFAR1 O14842 8/20 0.41
APEX1 P27695 1/20 0.40
FFAR4 Q5NUL3 5/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
HDAC3 O15379 1/20 0.37
MAPK1 P28482 1/20 0.37
ADRA1A P35348 1/20 0.37
HDAC4 P56524 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HDAC1 Q13547 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9632159 0.86 EGFR (0.36)
SCHEMBL5801660 0.70 KEAP1 (0.42) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL71453 0.69 PTGER4 (0.68) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL8484227 0.67 KEAP1 (0.50) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL59198 0.66 KEAP1 (0.65) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL31212507 0.65 PTGER4 (0.77) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL1261128 0.65 PTGER4 (0.77) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL6053663 0.63 PTGER4 (0.81) KEAP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL6535771 0.63 CDC25A (0.56) KEAP1FFAR1APEX1MEN1LMNA
SCHEMBL9264064 0.63 KEAP1 (0.46) KEAP1PTGER1PTGER4PTGER3PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2045483-A None JP disclosed
JP-2005247778-A METHOD FOR PRODUCING DIBENZOTHIEPINPROPIONIC ACID DERIVATIVE MAEKAWA SHIGEJI 2005-09-15 JP disclosed
JP-H0245483-A PREPARATION OF OPTICALLY ACTIVE DIBENZOTHIEPINPROPIONIC ACID NIPPON CHEMIPHAR CO LTD 1990-02-15 JP disclosed