SCHEMBL9632159

SCHEMBL9632159

NC(=O)CCC1=CSc2ccccc2-c2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
CAPN1 P07384 1/20 0.33
ATM Q13315 1/20 0.32
NR4A2 P43354 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PRMT1 Q99873 1/20 0.31
MTNR1A P48039 1/20 0.31
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6522978 0.86 KEAP1 (0.43)
SCHEMBL9321175 0.67 MTNR1A (0.47) EGFRSRCCAPN1NR4A2KDM4E
SCHEMBL9632170 0.65 MTNR1A (0.34) EGFRSRCATMMTNR1A
SCHEMBL6206188 0.65 PTGER4 (0.58) NR4A2
SCHEMBL3053811 0.64 TAAR1 (0.55) KDM4EMTNR1A
SCHEMBL30341383 0.64 TAAR1 (0.55) KDM4EMTNR1A
SCHEMBL20825056 0.62 SIGMAR1 (0.45) KDM4E
SCHEMBL27918771 0.62 MPO (0.50) ATMMTNR1A
SCHEMBL2593 0.62 KEAP1 (0.67) CAPN1PRMT1
Urea SCHEMBL6255302 0.61 KMT2A (0.50) SRCKDM4EBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0309626-B1 PROCESS FOR THE PREPARATION OF DIBENZOTHIEPIN DERIVATIVE NIPPON CHEMIPHAR CO., LTD. (JP) 1992-05-06 EP disclosed
US-4891433-A Process for the preparation of dibenzothiepin derivative NIPPON CHEMIPHAR CO., LTD. (JP) 1990-01-02 US disclosed
EP-0309626-A1 Process for the preparation of dibenzothiepin derivative NIPPON CHEMIPHAR CO., LTD. (JP) 1989-04-05 EP disclosed