SCHEMBL6526310

SCHEMBL6526310

O=S(=O)(O)c1ccccc1.OCCCN1CCc2ccccc2C1

nearest known ligand 0.65

Known targets — ChEMBL curated mechanism

BTKCACNA1CCACNA1DCACNA1FCACNA1SCACNA2D1CACNA2D2DRD2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQHRH1HTR2AP2RY12

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 3/20 0.58
DRD2 known ✓ P14416 3/20 0.56
HRH1 known ✓ P35367 1/20 0.56
HTR7 P34969 12/20 0.65
HTR1A P08908 4/20 0.58
DRD3 P35462 4/20 0.56
HTR2B P41595 2/20 0.56
SLC6A4 P31645 1/20 0.56
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
NCOR2 Q9Y618 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6521382 0.92 HTR7 (0.61) HTR7HTR1AHTR2ADRD3DRD2
SCHEMBL6521515 0.90 HTR7 (0.54) HTR7HTR1AHTR2ADRD3DRD2
SCHEMBL1828054 0.87 HTR1A (0.61) HTR7HTR1AHTR2ADRD3DRD2
SCHEMBL30305062 0.87 HTR1A (0.61) HTR7HTR1AHTR2ADRD3DRD2
Hydrochloric Acid SCHEMBL30541930 0.85 HTR1A (0.60) HTR7HTR1AHTR2ADRD3DRD2
Hydrochloric Acid SCHEMBL22527658 0.85 HTR1A (0.60) HTR7HTR1AHTR2ADRD3DRD2
Bromide SCHEMBL6523006 0.85 HTR1A (0.60) HTR7HTR1AHTR2ADRD3DRD2
Acetic Acid SCHEMBL6524435 0.85 DRD3 (0.64) HTR7HTR1AHTR2ADRD3DRD2
SCHEMBL6527411 0.82 USP2 (0.54) HTR7
SCHEMBL652976 0.80 HTR7 (0.60) HTR7HTR1AHTR2ADRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274056-B1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOCHINOLINIUM DERIVATIVES, SPECIFIC ALKANOLAMINES AND HYDROGEN PEROXYDE HENKEL AG & CO KGAA (DE) 2012-10-03 EP claimed
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE GROSS WIBKE 2011-03-10 US claimed
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE GROSS WIBKE 2011-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE KRT18, H1-3, H1-2 HTR2A 638/4885DRD2 791/4885HRH1 28/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.