SCHEMBL6532784

SCHEMBL6532784

O=C(C(O)CO)N1CCN(c2ccc(-n3cc(CN4C(=O)c5ccccc5C4=O)nn3)cc2F)CC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 1/20 0.41
ADRA1D P25100 3/20 0.40
ADRA1A P35348 3/20 0.40
ADRA1B P35368 3/20 0.40
PTGS2 P35354 5/20 0.38
GRM5 P41594 2/20 0.38
ALOX15 P16050 1/20 0.37
KCNH2 Q12809 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 1/20 0.35
TYR P14679 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532434 0.90 TYR (0.38) RBP4PTGS2ALOX15L3MBTL1HTT
SCHEMBL6533967 0.85 ADRA1D (0.42) ADRA1DADRA1AADRA1BPTGS2GRM5
SCHEMBL6529845 0.83 GPR119 (0.46) ADRA1DADRA1AADRA1BPTGS2GRM5
SCHEMBL5623713 0.81 ALDH1A1 (0.45) ADRA1DADRA1AADRA1BALOX15TYR
SCHEMBL6527396 0.79 ADRA1D (0.37) ADRA1DADRA1AADRA1BPTGS2ALOX15
SCHEMBL6532028 0.78 NOTUM (0.40) RBP4GRM5
SCHEMBL6527383 0.78 NOTUM (0.40) RBP4GRM5
SCHEMBL6532725 0.74 TYR (0.39) PTGS2ALOX15HTTTYR
SCHEMBL6534106 0.73 KDM1A (0.44) GRM5
SCHEMBL6532785 0.71 RBP4 (0.40) RBP4ADRA1DADRA1AADRA1BGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082892-A2 TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S LABORATORIES LTD. (IN) 2005-09-09 WO disclosed