SCHEMBL6533555

SCHEMBL6533555

COc1ccc(-c2ccccc2CCN(C(=O)C(C)Cl)c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
FFAR1 O14842 1/20 0.46
FFAR4 Q5NUL3 1/20 0.46
LPAR1 Q92633 3/20 0.43
LTB4R2 Q9NPC1 3/20 0.42
PPARA Q07869 3/20 0.41
CHRM5 P08912 2/20 0.41
CHRM1 P11229 2/20 0.41
CHRM3 P20309 2/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.39
MMP2 P08253 2/20 0.39
MMP9 P14780 2/20 0.39
MMP12 P39900 2/20 0.39
BACE1 P56817 1/20 0.39
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
MMP14 P50281 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533560 0.85 CHRM5 (0.53) ALDH1A1LPAR1CHRM5CHRM1CHRM3
SCHEMBL4938946 0.74 MTNR1A (0.51) ALDH1A1FFAR1FFAR4PPARA
SCHEMBL10896138 0.73 TP53 (0.43) ALDH1A1LTB4R2
SCHEMBL4216332 0.72 MMP2 (0.62) ALDH1A1FFAR1FFAR4LPAR1PTGDR2
SCHEMBL10900226 0.70 TSHR (0.39) ALDH1A1PPARA
SCHEMBL10987249 0.69 ALDH1A1 (0.50) ALDH1A1LTB4R2
SCHEMBL17940806 0.69 FFAR1 (0.56) FFAR1FFAR4LPAR1PPARAPTGDR2
SCHEMBL7596724 0.69 FFAR1 (0.52) FFAR1FFAR4PPARAPTGDR2MMP2
SCHEMBL6778364 0.68 PTGES (0.56) ALDH1A1LPAR1LTB4R2BACE1
SCHEMBL6716281 0.68 AOC3 (0.50) ALDH1A1CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005042491-A1 BENZAZEPINE DERIVATIVES AND METHODS OF PROPHYLAXIS OR TREATMENT OF 5HT2C RECEPTOR ASSOCIATED DISEASES ARENA PHARMACEUTICALS, INC. (US) 2005-05-12 WO disclosed