SCHEMBL6536056

SCHEMBL6536056

COC1=CC(C=O)(OCc2ccccc2)C(c2ccccc2)C=C1O

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ACHE P22303 1/20 0.32
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
FABP7 O15540 2/20 0.31
FABP5 Q01469 2/20 0.31
MIF P14174 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
LMNA P02545 1/20 0.31
MAOB P27338 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
AR P10275 1/20 0.30
RXRA P19793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6536233 0.88 ADORA3 (0.32) ALDH1A1TSHR
SCHEMBL6535991 0.76 KDM4E (0.33) KDM4EMAPTLMNAALDH1A1
SCHEMBL6536124 0.74 KDM4E (0.32) KDM4EMAPTLMNAALDH1A1SIRT1
SCHEMBL6536035 0.63 ERN1 (0.34) ERN1CYP2C9CYP2C19FABP7FABP5
SCHEMBL5215663 0.58 ALDH1A1 (0.30) ALDH1A1
SCHEMBL4752286 0.57 POLB (0.31)
Phenol SCHEMBL27648750 0.57 LMNA (0.54) CYP2C19MAPTLMNAMAOBALDH1A1
Phenol SCHEMBL28213971 0.57 LMNA (0.48) CYP2C9CYP2C19MIFLMNAALDH1A1
Phenol SCHEMBL27703621 0.55 CA12 (0.55) KDM4EMAPTALDH1A1TSHR
SCHEMBL14439823 0.55 TSHR (0.60) NPC1RAB9AKDM4EMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425015-A4 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-12-15 EP disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed