SCHEMBL6539459

SCHEMBL6539459

O=C(Nc1ccc(C[C@@H](CO)N(C[C@H](O)COc2ccccc2)C(=O)O)cc1)c1cccc2cccnc12

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
CASP3 P42574 1/20 0.46
RAB9A P51151 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
ADRB1 P08588 12/20 0.43
ADRB3 P13945 12/20 0.43
EGLN1 Q9GZT9 2/20 0.41
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6539444 0.88 KMT2A (0.52) ADRB1ADRB3ALDH1A1KMT2AITGB1
Hydrochloric Acid SCHEMBL6538979 0.82 ADRB3 (0.65) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL6539620 0.79 ADRB1 (0.46) NPC1RAB9AADRB1ADRB3MEN1
SCHEMBL6538847 0.79 ADRB1 (0.48) NPC1RAB9AADRB1ADRB3MEN1
SCHEMBL6539601 0.78 RAB9A (0.54) NPC1RAB9AADRB1ADRB3ALDH1A1
SCHEMBL6542153 0.78 MEN1 (0.48) NPC1RAB9AADRB1ADRB3MEN1
SCHEMBL6542157 0.78 MEN1 (0.48) NPC1RAB9AADRB1ADRB3MEN1
SCHEMBL6538911 0.78 ADRB3 (0.56) NPC1RAB9AADRB1ADRB3MEN1
SCHEMBL6538630 0.78 ADRB1 (0.43) ADRB1ADRB3POLBNPSR1
SCHEMBL6538698 0.77 NPC1 (0.43) NPC1RAB9AADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6826033-B2 BETA 3 ADRENERGIC RECEPTOR AGONISTS; TREATMENT OF POLLAKIURIA, URINARY INCONTINENCE, OBESITY OR DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-30 US disclosed
US-20040037022-A1 Aminoalcohol derivatives ASTELLAS PHARMA INC. (JP) 2004-02-26 US disclosed