Maleic Acid

Maleic Acid

SCHEMBL6544211

C1=CCC=C1.O=C(O)/C=C\C(=O)O

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
TP53 P04637 1/20 0.53
EGLN1 Q9GZT9 1/20 0.53
EGLN3 Q9H6Z9 1/20 0.53
HCAR2 Q8TDS4 4/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 5/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 2/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C9 P11712 1/20 0.34
HTT P42858 2/20 0.33
HDAC3 O15379 1/20 0.33
TNKS O95271 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL16099816 1.00 TSHR (0.53) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL958116 1.00 TSHR (0.53) TSHRTP53EGLN1EGLN3HCAR2
Maleic Acid SCHEMBL9580936 1.00 TSHR (0.53) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL27903060 0.97 TSHR (0.50) TSHRTP53EGLN1EGLN3HCAR2
Monomethyl Fumarate SCHEMBL28979771 0.82 HCAR2 (0.68) TSHRTP53EGLN1EGLN3HCAR2
Monomethyl Fumarate SCHEMBL11141023 0.82 HCAR2 (0.68) TSHRTP53EGLN1EGLN3HCAR2
Bicarbonate SCHEMBL6249355 0.81 CA1 (0.39)
Bicarbonate SCHEMBL7515371 0.81 CA1 (0.39)
Bicarbonate SCHEMBL9418217 0.81
Bicarbonate SCHEMBL283948 0.81 CA1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118725422-A Carcass rubber composition for reducing carbon black use, preparation method thereof and tire 中策橡胶集团股份有限公司 2024-10-01 CN claimed
CN-118599194-A Tire transition layer rubber composition for reducing carbon black use, preparation method thereof and tire 中策橡胶集团股份有限公司 2024-09-06 CN claimed
CN-114478840-B Functionalized reversion liquid rubber and preparation method thereof 杭州中策橡胶循环科技有限公司 2022-09-06 CN claimed
CN-114478840-A Functionalized reversion liquid rubber and preparation method thereof 杭州中策橡胶循环科技有限公司 2022-05-13 CN claimed
EP-2976380-B1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY Henkel IP & Holding GmbH (DE) 2018-10-10 EP claimed
US-20180155588-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY HENKEL AG & CO. KGAA (DE) 2018-06-07 US claimed
US-9938437-B2 Diene/dienophile couples and thermosetting resin compositions having reworkability Henkel IP & Holding GmbH (DE) 2018-04-10 US claimed
EP-2976380-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY Henkel IP & Holding GmbH (DE) 2016-01-27 EP claimed
US-20160002510-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY HENKEL AG & CO. KGAA (DE) 2016-01-07 US claimed
WO-2014153513-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY Henkel IP & Holding GmbH (DE) 2014-09-25 WO claimed
CN-118725422-A Carcass rubber composition for reducing carbon black use, preparation method thereof and tire 中策橡胶集团股份有限公司 2024-10-01 CN disclosed
CN-118599194-A Tire transition layer rubber composition for reducing carbon black use, preparation method thereof and tire 中策橡胶集团股份有限公司 2024-09-06 CN disclosed
CN-114478840-B Functionalized reversion liquid rubber and preparation method thereof 杭州中策橡胶循环科技有限公司 2022-09-06 CN disclosed
CN-114478840-A Functionalized reversion liquid rubber and preparation method thereof 杭州中策橡胶循环科技有限公司 2022-05-13 CN disclosed
CN-107365400-B A kind of synthetic method of styrene-dicyclopentadiene monomaleate copolymer 中国科学院新疆理化技术研究所 2019-11-19 CN disclosed
WO-2014153513-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY Henkel IP & Holding GmbH (DE) 2014-09-25 WO disclosed
CN-102407633-A Combined Lamination Body JSP K K 2012-04-11 CN disclosed
US-20040116643-A1 Composite resin and use thereof TOYO INK MFG. CO., LTD. (JP) 2004-06-17 US disclosed
EP-1375558-A1 COMPOSITE RESIN AND USE THEREOF TOYO INK MFG. CO., LTD. (JP) 2004-01-02 EP disclosed
US-4105607-A COPOLYMER OF DICYCLOPENTADIENE AND AN OLEFINICALLY UNSATURATED CARBOXYLIC ACID OR ALCOHOL HOECHST AKTIENGESELLSCHAFT (DE) 1978-08-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160002510-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY GCN1, GSS, LSS TSHR 4372/4885TP53 4004/4885EGLN1 1905/4885
US-20180155588-A1 DIENE/DIENOPHILE COUPLES AND THERMOSETTING RESIN COMPOSITIONS HAVING REWORKABILITY GCN1, GSS, LSS TSHR 4372/4885TP53 4004/4885EGLN1 1905/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.