SCHEMBL655212

SCHEMBL655212

C=CCN(CC=C)c1ccccc1C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.46
PTPN1 P18031 1/20 0.44
ALDH1A1 P00352 6/20 0.41
TSHR P16473 3/20 0.41
HPGD P15428 3/20 0.41
MAPT P10636 3/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP3A4 P08684 1/20 0.40
METAP2 P50579 1/20 0.39
BCAT2 O15382 1/20 0.38
PARP1 P09874 1/20 0.37
HTT P42858 1/20 0.37
ALOX5 P09917 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.36
C5AR1 P21730 1/20 0.36
GAA P10253 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL89548 0.86 ALDH1A1 (0.50) KDM4EPTPN1ALDH1A1TSHRHPGD
SCHEMBL278676 0.84 PTPN1 (0.47) KDM4EPTPN1ALDH1A1TSHRHPGD
SCHEMBL11120806 0.83 KDM4E (0.38) KDM4EPTPN1ALDH1A1TSHRHPGD
Hydrochloric Acid SCHEMBL27897977 0.83 PTPN1 (0.46) KDM4EPTPN1ALDH1A1TSHRHPGD
SCHEMBL21084683 0.83 PTPN1 (0.44) KDM4EPTPN1ALDH1A1TSHRHPGD
SCHEMBL10692029 0.80 PTPN1 (0.43) KDM4EPTPN1ALDH1A1TSHRHPGD
SCHEMBL83996 0.80 AKR1C3 (0.46) PTPN1ALDH1A1TSHRHPGDMAPT
Benzophenone SCHEMBL27852184 0.79 ALDH1A1 (0.45) PTPN1ALDH1A1TSHRHPGDMAPT
SCHEMBL11767364 0.79 AKR1C3 (0.44) KDM4EPTPN1ALDH1A1TSHRMAPT
SCHEMBL8946208 0.79 CYP1A2 (0.41) KDM4EPTPN1ALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0738138-A1 QUATERNARY SALTS OF PARA-DIALKYLAMINO BENZAMIDE DERIVATIVES ISP Van Dyk Inc. (US) 1996-10-23 EP claimed
EP-0738138-A4 QUATERNARY SALTS OF PARA-DIALKYLAMINO BENZAMIDE DERIVATIVES ISP VAN DYK INC (US) 1996-07-08 EP claimed
WO-1995005797-A1 QUATERNARY SALTS OF PARA-DIALKYLAMINO BENZAMIDE DERIVATIVES ISP VAN DYK INC. (US) 1995-03-02 WO claimed
CN-109180394-A A kind of granular urea preparation method containing alginic acid synergistic carrier suitable for winter wheat top dressing 中国农业科学院农业资源与农业区划研究所 2019-01-11 CN disclosed
EP-2013196-B1 DISUBSTITUTED ANILINE COMPOUNDS MERCK SHARP & DOHME (US) 2015-09-16 EP disclosed
US-8119685-B2 Disubstituted aniline compounds MERCK SHARP & DOHME CORP. (US) 2012-02-21 US disclosed
US-20090221669-A1 Disubstituted Aniline Compounds MERCK SHARP & DOHME LLC 2009-09-03 US disclosed
EP-2013196-A2 DISUBSTITUTED ANILINE COMPOUNDS Merck & Co., Inc. (US) 2009-01-14 EP disclosed
WO-2007127137-A2 DISUBSTITUTED ANILINE COMPOUNDS MERCK & CO., INC. (US) 2007-11-08 WO disclosed
US-5427773-A Sunscreen agents ISP VAN DYK INC. (US) 1995-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090221669-A1 Disubstituted Aniline Compounds TXNRD2, BRDT, HDAC1 KDM4E 500/4885PTPN1 1085/4885ALDH1A1 744/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.