SCHEMBL6559026

SCHEMBL6559026

CC(=O)OC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)[C@@H](O)[C@@H](O)[C@H](O)C(=O)N[C@@H](CC(=O)O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.48
CTSB P07858 5/20 0.48
PSMB1 P20618 1/20 0.48
REN P00797 2/20 0.46
CTSD P07339 1/20 0.44
CASP3 P42574 3/20 0.44
CASP7 P55210 2/20 0.43
CTSS P25774 3/20 0.43
CTSL P07711 3/20 0.43
CASP1 P29466 1/20 0.43
CASP4 P49662 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559234 0.92 CTSK (0.50) CTSKCTSBPSMB1RENCTSD
SCHEMBL6559868 0.85 PSMB1 (0.39) PSMB1RENCTSD
SCHEMBL6558995 0.85 PSMB1 (0.56) CTSKCTSBPSMB1CTSSCTSL
SCHEMBL6560838 0.83 CTSK (0.52) CTSKCTSBPSMB1RENCTSS
SCHEMBL6558612 0.79 PSMB1 (0.50) CTSKCTSBPSMB1RENCTSS
SCHEMBL6564394 0.79 PSMB1 (0.50) CTSKCTSBPSMB1CTSSCTSL
SCHEMBL6560880 0.79 PSMB1 (0.64) CTSKCTSBPSMB1CTSSCTSL
SCHEMBL6558606 0.78 PSMB1 (0.43) CTSKPSMB1RENCTSDCTSS
SCHEMBL7741834 0.78 CASP3 (0.40) CTSDCASP3CASP7CASP1
SCHEMBL6559358 0.77 CTSD (0.45) CTSDCASP3CASP7CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998488-B1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-03-17 EP disclosed
US-6423869-B1 BACTERICIDES, ANTIULCER AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-07-23 US disclosed