SCHEMBL6559970

SCHEMBL6559970

Nc1ccc(S(=O)(=O)N2CCC(=O)C2)cc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.56
MMP2 P08253 1/20 0.54
PKM P14618 5/20 0.49
MEN1 O00255 3/20 0.46
AKR1C3 P42330 3/20 0.45
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
NT5E P21589 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557849 0.89 USP2 (0.53) KMT2AMMP2PKMMEN1AKR1C3
SCHEMBL265611 0.83 PKM (0.61) KMT2AMMP2PKMMEN1ALDH1A1
SCHEMBL11306227 0.79 PKM (0.69) KMT2AMMP2PKMMEN1USP2
SCHEMBL2299332 0.79 KMT2A (0.51) KMT2APKMMEN1AKR1C3USP2
SCHEMBL20389408 0.79 KMT2A (0.77) KMT2AMEN1AKR1C3ALDH1A1TSHR
SCHEMBL3637211 0.79 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1
SCHEMBL8218091 0.77 PKM (0.54) KMT2AMMP2PKMMEN1USP2
SCHEMBL14132273 0.76 MCOLN3 (0.55) KMT2APKMMEN1AKR1C3USP2
SCHEMBL78283 0.76 USP2 (0.69) KMT2AMMP2PKMMEN1USP2
SCHEMBL655768 0.76 USP2 (0.76) KMT2APKMMEN1USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436255-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS Aventis Pharmaceuticals, Inc. (US) 2004-07-14 EP disclosed
WO-2003024924-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2003-03-27 WO disclosed