SCHEMBL265611

SCHEMBL265611

Cc1ccc(S(=O)(=O)N2CCC(=O)C2)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.61
HTT P42858 2/20 0.59
ALDH1A1 P00352 1/20 0.59
POLB P06746 1/20 0.59
CD4 P01730 5/20 0.57
KMT2A Q03164 4/20 0.56
MMP2 P08253 1/20 0.54
MEN1 O00255 3/20 0.54
GAA P10253 2/20 0.54
TSHR P16473 1/20 0.54
CYP2C19 P33261 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
LMNA P02545 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12169347 0.90 PKM (0.65) PKMHTTALDH1A1POLBCD4
SCHEMBL2448500 0.89 PKM (0.70) PKMHTTALDH1A1POLBKMT2A
SCHEMBL505093 0.89 KMT2A (0.69) PKMHTTALDH1A1POLBKMT2A
SCHEMBL17369299 0.89 PKM (0.64) PKMHTTALDH1A1POLBKMT2A
SCHEMBL11605844 0.85 PKM (0.63) PKMHTTALDH1A1POLBKMT2A
SCHEMBL6559970 0.83 KMT2A (0.56) PKMALDH1A1KMT2AMMP2MEN1
SCHEMBL12330050 0.83 PKM (0.61) PKMHTTALDH1A1POLBCD4
SCHEMBL8024905 0.82 KMT2A (0.64) PKMHTTALDH1A1POLBKMT2A
SCHEMBL9693041 0.80 PKM (0.66) PKMHTTALDH1A1POLBKMT2A
SCHEMBL4537086 0.79 PKM (0.88) PKMHTTALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190321313-A1 BENZENESULFONAMIDE DERIVATIVES AND METHOD FOR TREATING CANCER Gongwin Biopharm Holdings Co., Ltd. 2019-10-24 US disclosed
US-9782370-B2 Pharmaceutical compositions of benzenesulfonamide derivatives for treatment of adenoid cystic carcinoma Gongwin Biopharm Holdings Co., Ltd. (KY) 2017-10-10 US disclosed
US-20170172951-A1 NOVEL PHARMACEUTICAL COMPOSITIONS OF BENZENESULFONAMIDE DERIVATIVES FOR TREATMENT OF ADENOID CYSTIC CARCINOMA GONGWIN BIOPHARM CO., LTD. (TAIWAN) (TW) 2017-06-22 US disclosed
US-8431378-B2 Aminotransferase, gene encoding the same, and methods of using them KANEKA CORPORATION (JP) 2013-04-30 US disclosed
US-20120164724-A1 NOVEL AMINOTRANSFERASE, GENE ENCODING THE SAME, AND METHODS OF USING THEM KANEKA CORPORATION (JP) 2012-06-28 US disclosed
US-8133705-B2 Aminotransferase, gene encoding the same, and method of using them KANEKA CORPORATION (JP) 2012-03-13 US disclosed
US-8039467-B2 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION (US) 2011-10-18 US disclosed
US-8039467-B2 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION (US) 2011-10-18 US disclosed
US-20100285544-A1 Novel aminotransferase, gene encoding the same, and method of using them KANEKA CORPORATION (JP) 2010-11-11 US disclosed
US-20100145048-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS SCHERING CORPORATION 2010-06-10 US disclosed
US-7638513-B2 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION (US) 2009-12-29 US disclosed
US-7638513-B2 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION (US) 2009-12-29 US disclosed
EP-1889907-B1 NOVEL AMINO GROUP TRANSFERASE, GENE ENCODING THE SAME AND METHOD OF USING THE SAME KANEKA CORP (JP) 2009-09-02 EP disclosed
EP-1889907-A1 NOVEL AMINO GROUP TRANSFERASE, GENE ENCODING THE SAME AND METHOD OF USING THE SAME Kaneka Corporation (JP) 2008-02-20 EP disclosed
US-20070167426-A1 Compounds for the treatment of inflammatory disorders and microbial diseases SCHERING CORPORATION 2007-07-19 US disclosed
US-20070167426-A1 Compounds for the treatment of inflammatory disorders and microbial diseases SCHERING CORPORATION 2007-07-19 US disclosed
WO-2007064749-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS AND MICROBIAL DISEASES SCHERING CORPORATION (US) 2007-06-07 WO disclosed
US-20060178366-A1 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION 2006-08-10 US disclosed
US-20060178366-A1 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION 2006-08-10 US disclosed
WO-2005121130-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR THE TREATMENT OF INFLAMMATORY DISORDERS SCHERING CORPORATION (US) 2005-12-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167426-A1 Compounds for the treatment of inflammatory disorders and microbial diseases MMP12, ADAMTS1, ADAM33 PKM 2433/4885HTT 1008/4885ALDH1A1 1502/4885
US-20190321313-A1 BENZENESULFONAMIDE DERIVATIVES AND METHOD FOR TREATING CANCER ARSA, ABCB1, ABCG2 PKM 1749/4885HTT 902/4885ALDH1A1 689/4885
US-20170172951-A1 NOVEL PHARMACEUTICAL COMPOSITIONS OF BENZENESULFONAMIDE DERIVATIVES FOR TREATMENT OF ADENOID CYSTIC CARCINOMA ABCD3, CFTR, ADSL PKM 3549/4885HTT 2849/4885ALDH1A1 1243/4885
US-20060178366-A1 Compounds for the treatment of inflammatory disorders MMP12, ADAMTS1, TNF PKM 2167/4885HTT 1281/4885ALDH1A1 1369/4885
US-20100145048-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS TNF, MMP12, MMP8 PKM 2069/4885HTT 1719/4885ALDH1A1 1342/4885
US-20100285544-A1 Novel aminotransferase, gene encoding the same, and method of using them BCAT1, AGXT, ALDH7A1 PKM 424/4885HTT 2680/4885ALDH1A1 144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.