SCHEMBL6560132

SCHEMBL6560132

COc1cc(N[C]=O)cc(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
KMT2A Q03164 3/20 0.46
POLB P06746 1/20 0.46
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TP53 P04637 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
GAA P10253 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.42
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5457581 0.82 HDAC3 (0.47) AKR1C3AKR1C2MAPT
SCHEMBL1188677 0.79 KMT2A (0.56) ALDH1A1KMT2APOLBRAB9ANPC1
SCHEMBL225906 0.77 RAB9A (0.56) ALDH1A1RAB9ANPC1SMN1; SMN2TP53
SCHEMBL2092658 0.74 ACHE (0.52) ALDH1A1KMT2APOLBSMN1; SMN2MEN1
SCHEMBL3557737 0.74 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2TP53CYP1A2CYP3A4
SCHEMBL3555814 0.72 CYP3A4 (0.48) ALDH1A1POLBRAB9ANPC1SMN1; SMN2
SCHEMBL3188883 0.72 ALDH1A1 (0.65) ALDH1A1KMT2APOLBRAB9ANPC1
1,3,5-Trimethoxybenzene SCHEMBL28493 0.71 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1547868 0.70 ALDH1A1 (0.61) ALDH1A1KMT2APOLBRAB9ANPC1
SCHEMBL424460 0.70 RAPGEF4 (0.42) ALDH1A1KMT2AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-1146865-B9 PHARMACEUTICAL COMPOSITION COMPRISING A COMBINATION OF DEXTRO- AND LAEVO- ISOMERS OF SOTALOL TORRENT PHARMACEUTICALS LTD (IN) 2004-03-17 EP disclosed
EP-1146865-B1 PHARMACEUTICAL COMPOSITION COMPRISING A COMBINATION OF DEXTRO- AND LAEVO- ISOMERS OF SOTALOL TORRENT PHARMACEUTICALS LTD (IN) 2003-05-28 EP disclosed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
EP-1146865-A1 PHARMACEUTICAL COMPOSITION COMPRISING A COMBINATION OF DEXTRO- AND LAEVO- ISOMERS OF SOTALOL Torrent Pharmaceuticals Ltd (IN) 2001-10-24 EP disclosed
US-6281246-B2 CONTROLLING RATIOS OF ISOMERS TORRENT PHARMACEUTICAL LTD. (IN) 2001-08-28 US disclosed
US-20010004643-A1 Pharmaceutical composition with sotalol combination and their use in treatment of cardiac ailments THE ROSHNI SINGH 2015 TRUST 2001-06-21 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed
WO-2000045807-A1 PHARMACEUTICAL COMPOSITION COMPRISING A COMBINATION OF DEXTRO- AND LAEVO- ISOMERS OF SOTALOL SANKARANARAYANAN ALANGUDI (IN) 2000-08-10 WO disclosed
US-5939398-A ANTIATHEROSCLEROSIS AGENTS PFIZER INC. (US) 1999-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010004643-A1 Pharmaceutical composition with sotalol combination and their use in treatment of cardiac ailments ADRB1, ADRB2, ADRB3 ALDH1A1 525/4885KMT2A 4204/4885POLB 2097/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.