SCHEMBL6561655

SCHEMBL6561655

Nc1ccccc1NS(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.77

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.66
TSHR P16473 1/20 0.66
KMT2A Q03164 1/20 0.66
KEAP1 Q14145 1/20 0.65
NFE2L2 Q16236 1/20 0.65
PKM P14618 1/20 0.55
MCOLN3 Q8TDD5 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CHEK1 O14757 1/20 0.52
CDK8 P49336 1/20 0.52
NEK2 P51955 1/20 0.52
LIMK1 P53667 1/20 0.52
GLO1 Q04760 1/20 0.52
STAT3 P40763 1/20 0.52
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30737629 1.00 MEN1 (0.66) MEN1TSHRKMT2AKEAP1NFE2L2
SCHEMBL7589375 0.87 MEN1 (0.77) MEN1TSHRKMT2AKEAP1NFE2L2
SCHEMBL2068236 0.85 ALDH1A1 (0.58) MEN1KMT2AKEAP1PKMGLO1
SCHEMBL30737452 0.85 ALDH1A1 (0.58) MEN1KMT2AKEAP1PKMGLO1
Hydrochloric Acid SCHEMBL29885455 0.84 ALDH1A1 (0.56) MEN1KMT2AKEAP1PKMGLO1
SCHEMBL30737499 0.83 ALDH1A1 (0.66) MEN1TSHRKMT2A
SCHEMBL398000 0.83 LMNA (0.70) MEN1TSHRKMT2AKEAP1NFE2L2
SCHEMBL15145878 0.83 MEN1 (0.52) MEN1KMT2AL3MBTL1
SCHEMBL4184006 0.83 ALDH1A1 (0.66) MEN1TSHRKMT2A
SCHEMBL7854392 0.82 TSHR (0.70) MEN1TSHRKMT2AKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117510460-A Benzo [ b ] thiophene derivative containing sulfonamide unit, and preparation method and application thereof 贵州大学 2024-02-06 CN disclosed
US-9216954-B2 Serine racemase inhibitor NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2015-12-22 US disclosed
US-9216954-B2 Serine racemase inhibitor NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2015-12-22 US disclosed
US-20140371291-A1 SERINE RACEMASE INHIBITOR NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2014-12-18 US disclosed
US-20140371291-A1 SERINE RACEMASE INHIBITOR NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2014-12-18 US disclosed
EP-2808014-A1 SERINE RACEMASE INHIBITOR National University Corporation University Of Toyama (JP) 2014-12-03 EP disclosed
EP-2808014-A1 SERINE RACEMASE INHIBITOR National University Corporation University Of Toyama (JP) 2014-12-03 EP disclosed
WO-2013111798-A1 SERINE RACEMASE INHIBITOR 国立大学法人 富山大学 (JP) 2013-08-01 WO disclosed
EP-0990645-B1 NOVEL SULFONAMIDE DERIVATIVES NIPPON KAYAKU KK (JP) 2004-07-28 EP disclosed
US-6458960-B1 ANTICANCER AGENTS, RHEUMATIC DISEASES AND ANTIINFLAMMATORY AGENTS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2002-10-01 US disclosed
US-6180796-B1 TUBULIN POLYMERIZATION INHIBITORS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-01-30 US disclosed
EP-0990645-A1 NOVEL SULFONAMIDE DERIVATIVES Nippon Kayaku Kabushiki Kaisha (JP) 2000-04-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140371291-A1 SERINE RACEMASE INHIBITOR SRR, PRSS1, ME1 MEN1 1089/4885TSHR 4233/4885KMT2A 3922/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.