SCHEMBL6561733

SCHEMBL6561733

COc1ccc(S(=O)(=O)Nc2ccccc2NC(=O)c2c(-c3ccccc3)noc2C)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.64
ALDH1A1 P00352 8/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
LMNA P02545 4/20 0.56
KDM4E B2RXH2 4/20 0.56
KMT2A Q03164 3/20 0.56
HPGD P15428 2/20 0.56
HSD17B10 Q99714 2/20 0.56
MEN1 O00255 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
POLB P06746 2/20 0.56
GAA P10253 1/20 0.56
CRHBP P24387 1/20 0.56
CRHR2 Q13324 1/20 0.56
PKM P14618 1/20 0.55
ALOX12 P18054 1/20 0.55
HTT P42858 1/20 0.55
TP53 P04637 1/20 0.54
MAPT P10636 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6562122 0.88 ALOX15 (0.54) TSHRALDH1A1L3MBTL1LMNAKDM4E
SCHEMBL6563188 0.84 KEAP1 (0.49) TSHRALDH1A1L3MBTL1LMNAKDM4E
SCHEMBL6563185 0.84 TDP1 (0.53) ALDH1A1L3MBTL1LMNAKDM4EKMT2A
SCHEMBL6563164 0.78 ALDH1A1 (0.54) ALDH1A1L3MBTL1LMNAKDM4EKMT2A
SCHEMBL6561737 0.78 KEAP1 (0.49) TSHRALDH1A1L3MBTL1LMNAKDM4E
SCHEMBL6561650 0.78 KEAP1 (0.53) TSHRALDH1A1L3MBTL1LMNAKDM4E
SCHEMBL8625192 0.77 F10 (0.67) ALDH1A1L3MBTL1LMNAKDM4EKMT2A
SCHEMBL6561679 0.77 ALDH1A1 (0.49) ALDH1A1L3MBTL1LMNAKDM4EKMT2A
SCHEMBL328337 0.76 ALDH1A1 (0.74) TSHRALDH1A1L3MBTL1LMNAKDM4E
SCHEMBL8626109 0.76 CCR9 (0.66) KMT2AHPGDMEN1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0990645-B1 NOVEL SULFONAMIDE DERIVATIVES NIPPON KAYAKU KK (JP) 2004-07-28 EP disclosed
US-6180796-B1 TUBULIN POLYMERIZATION INHIBITORS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-01-30 US disclosed
EP-0990645-A1 NOVEL SULFONAMIDE DERIVATIVES Nippon Kayaku Kabushiki Kaisha (JP) 2000-04-05 EP disclosed