SCHEMBL6561679

SCHEMBL6561679

CCc1noc(CC)c1C(=O)Nc1ccccc1NS(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
LMNA P02545 3/20 0.49
TP53 P04637 2/20 0.49
HPGD P15428 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HTT P42858 1/20 0.49
HDAC3 O15379 3/20 0.48
HDAC1 Q13547 3/20 0.48
NCOR2 Q9Y618 3/20 0.48
HDAC2 Q92769 2/20 0.48
KEAP1 Q14145 2/20 0.46
KCNA5 P22460 1/20 0.46
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46
TUBA3C P0DPH7 1/20 0.46
TUBA1B P68363 1/20 0.46
TUBA4A P68366 1/20 0.46
TUBB4B P68371 1/20 0.46
TUBB3 Q13509 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563185 0.90 TDP1 (0.53) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6563164 0.90 ALDH1A1 (0.54) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6561743 0.81 LMNA (0.53) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6562122 0.80 ALOX15 (0.54) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6563188 0.77 KEAP1 (0.49) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6561737 0.77 KEAP1 (0.49) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6561733 0.77 TSHR (0.64) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL8625192 0.75 F10 (0.67) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL6561650 0.73 KEAP1 (0.53) ALDH1A1L3MBTL1LMNATP53HPGD
SCHEMBL8626468 0.73 SMN1; SMN2 (0.69) ALDH1A1L3MBTL1LMNASMN1; SMN2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0990645-B1 NOVEL SULFONAMIDE DERIVATIVES NIPPON KAYAKU KK (JP) 2004-07-28 EP disclosed
US-6180796-B1 TUBULIN POLYMERIZATION INHIBITORS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-01-30 US disclosed
EP-0990645-A1 NOVEL SULFONAMIDE DERIVATIVES Nippon Kayaku Kabushiki Kaisha (JP) 2000-04-05 EP disclosed