SCHEMBL6561930

SCHEMBL6561930

CCOC(=O)CN(C)Cc1cc(C#CCNc2ccccc2)ccc1C(=O)N1CCCC1C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 1/20 0.39
TP53 P04637 1/20 0.37
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KCNK3 O14649 8/20 0.34
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
HTT P42858 2/20 0.34
NAMPT P43490 1/20 0.34
ITGB2 P05107 1/20 0.34
ICAM1 P05362 1/20 0.34
ITGAL P20701 1/20 0.34
MAP3K7 O43318 1/20 0.32
TAB1 Q15750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7671224 0.90 PRSS1 (0.35) MEN1KMT2ATSHRALDH1A1SMN1; SMN2
SCHEMBL6561843 0.85 GAA (0.31) MEN1KMT2ATSHRSMN1; SMN2NAMPT
SCHEMBL7669679 0.81 F2 (0.37) MEN1KMT2AMAPK1ALDH1A1HTT
SCHEMBL6563261 0.72 HSD11B1 (0.38) ALDH1A1MAPTHTTNAMPT
SCHEMBL6565512 0.71 GAA (0.40) MEN1KMT2AMAPK1ALDH1A1NAMPT
SCHEMBL7804851 0.70 HRH3 (0.36)
SCHEMBL7806152 0.69 HRH3 (0.37) ALDH1A1
SCHEMBL6561835 0.69 PTPN11 (0.35) MEN1KMT2AALDH1A1MAPTKCNK3
SCHEMBL6563696 0.68 HPGD (0.37) MEN1KMT2ATSHRKDM4EALDH1A1
SCHEMBL6565856 0.68 IMPDH2 (0.38) MEN1KMT2ATSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed