SCHEMBL6563591

SCHEMBL6563591

COc1cc(C(=O)N2CCCC2C)ccc1C#CCNc1ccc(C(=N)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.39
ROCK2 O75116 2/20 0.38
HSD11B1 P28845 3/20 0.37
GAA P10253 2/20 0.35
HPGD P15428 1/20 0.35
NAMPT P43490 1/20 0.35
HTT P42858 1/20 0.35
HRH3 Q9Y5N1 2/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.34
RORC P51449 1/20 0.34
TLR8 Q9NR97 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
MEN1 O00255 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
PDK2 Q15119 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563605 0.91 GAA (0.37) HSD11B1GAAHPGDNAMPTHTT
SCHEMBL6563002 0.86 HRH3 (0.42) HSD11B1GAAHPGDNAMPTHRH3
SCHEMBL6563266 0.85 LRRK2 (0.42) LRRK2ROCK2HSD11B1GAAHPGD
SCHEMBL6563752 0.85 GAA (0.35) HSD11B1GAAHPGDNAMPTHTT
SCHEMBL6565417 0.84 PTPN11 (0.36) HSD11B1GAAHPGDNAMPTHRH3
SCHEMBL6561835 0.82 PTPN11 (0.35) HSD11B1GAAHPGDNAMPTHTT
SCHEMBL6563507 0.79 KCNK3 (0.31) HSD11B1GAAHPGDNAMPTHTT
SCHEMBL6563920 0.78 KLK5 (0.41) ROCK2ALDH1A1KMT2APDK2
SCHEMBL6563568 0.77 CNR2 (0.39) GAAHPGDNAMPTHTTPOLB
SCHEMBL6563511 0.77 PTPN11 (0.40) ROCK2HSD11B1POLBPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed