SCHEMBL6566003

SCHEMBL6566003

CC1CCCN1C(=O)c1cc(Br)c(C#CCNc2ccc(C(=N)N)cc2)o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 5/20 0.37
GAA P10253 2/20 0.37
HPGD P15428 2/20 0.37
F10 P00742 1/20 0.37
PRSS1 P07477 1/20 0.37
ADORA2A P29274 3/20 0.37
NAMPT P43490 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561857 0.86 F2 (0.43) F2F10PRSS1ALDH1A1NPC1
SCHEMBL6561970 0.81 GAA (0.49) F2GAAHPGDNAMPTCA12
SCHEMBL6563410 0.80 GAA (0.40) F2GAAHPGDF10PRSS1
SCHEMBL6565356 0.79 GAA (0.42) F2GAAHPGDF10PRSS1
SCHEMBL6565512 0.79 GAA (0.40) F2GAAHPGDF10PRSS1
SCHEMBL6563266 0.77 LRRK2 (0.42) GAAHPGDNAMPTCA12CA1
SCHEMBL6563261 0.76 HSD11B1 (0.38) F2GAAHPGDF10PRSS1
SCHEMBL6564299 0.73 GAA (0.36) F2GAAHPGDF10PRSS1
SCHEMBL7669679 0.73 F2 (0.37) F2GAAHPGDF10PRSS1
SCHEMBL6561673 0.71 PRSS1 (0.35) F2GAAHPGDF10PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed