SCHEMBL6563328

SCHEMBL6563328

CC(C)(C)OC(=O)NC(=N)c1ccc(NCC#Cc2ccc(C(=O)N3CCCC3)c(C=O)c2)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.36
PTPN11 Q06124 1/20 0.35
ABL1 P00519 1/20 0.34
RIN1 Q13671 1/20 0.34
CNR2 P34972 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
HSD11B1 P28845 1/20 0.32
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31
F10 P00742 1/20 0.31
JAK1 P23458 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
SPIN1 Q9Y657 1/20 0.30
ACHE P22303 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565533 0.90 ACACB (0.45) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL6561810 0.89 HSD11B1 (0.40) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL6565339 0.89 HPGD (0.39) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL7674981 0.86 ABL1 (0.43) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL7686729 0.84 PTPN11 (0.43) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL6565093 0.84 ACACB (0.35) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL6563597 0.84 F10 (0.38) ACACBF10
SCHEMBL6561973 0.83 JAK1 (0.38) ACACBPTPN11JAK1KMT2A
SCHEMBL6563912 0.83 ACACB (0.34) ACACBPTPN11ABL1RIN1CNR2
SCHEMBL6565336 0.83 ACACB (0.34) ACACBPTPN11ABL1RIN1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed