SCHEMBL6563680

SCHEMBL6563680

COc1cc(C(=N)N)ccc1NCC#Cc1ccc(C(=O)c2ccccc2)c(C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.40
GAA P10253 2/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 5/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 3/20 0.39
HTT P42858 1/20 0.39
PDE5A O76074 1/20 0.39
ABCC9 O60706 1/20 0.38
ABCC8 Q09428 1/20 0.38
KCNJ11 Q14654 1/20 0.38
KCNJ8 Q15842 1/20 0.38
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 2/20 0.37
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PRSS1 P07477 3/20 0.37
ASIC3 Q9UHC3 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565231 0.86 GAA (0.41) PPARGGAATP53MAPTSMN1; SMN2
SCHEMBL6563277 0.84 F2 (0.41) PRSS1ASIC3PLAUKLK1KLK5
SCHEMBL6563737 0.78 EGLN1 (0.45) GAALMNAKDM4EL3MBTL1HPGD
SCHEMBL7675063 0.73 F2 (0.48) PRSS1PLAUKLK1KLK5
SCHEMBL6563213 0.73 KMT2A (0.39) MAPTPRSS1PLAU
SCHEMBL5885884 0.72 PTPN1 (0.39) L3MBTL1PRSS1ASIC3PLAU
SCHEMBL6563625 0.71 PRSS1 (0.43) LMNAL3MBTL1PRSS1ASIC3HPGD
Hydrochloric Acid SCHEMBL5885907 0.71 PTPN1 (0.39) L3MBTL1PRSS1ASIC3PLAU
SCHEMBL5885889 0.70 F10 (0.38) PRSS1ASIC3
SCHEMBL6563946 0.69 KLK1 (0.42) SMN1; SMN2PRSS1HPGDPLAUKLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed