SCHEMBL6563752

SCHEMBL6563752

Cc1cc(C(=O)N2CCCC2C)c(C)cc1C#CCNc1ccc(C(=N)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 2/20 0.34
NAMPT P43490 1/20 0.34
NPC1 O15118 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
HSD11B1 P28845 1/20 0.34
KCNK3 O14649 4/20 0.33
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HTT P42858 1/20 0.32
TSHR P16473 1/20 0.32
RORC P51449 1/20 0.32
RORB Q92753 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563605 0.91 GAA (0.37) GAAALDH1A1HPGDNAMPTNPC1
SCHEMBL6563507 0.90 KCNK3 (0.31) GAAALDH1A1HPGDNAMPTNPC1
SCHEMBL6565417 0.90 PTPN11 (0.36) GAAALDH1A1HPGDNAMPTNPC1
SCHEMBL6561938 0.87 ABL1 (0.36) GAAALDH1A1HPGDMEN1KMT2A
SCHEMBL6563627 0.86 PTPN11 (0.33)
SCHEMBL6563002 0.85 HRH3 (0.42) GAAALDH1A1HPGDNAMPTNPC1
SCHEMBL6563591 0.85 LRRK2 (0.39) GAAALDH1A1HPGDNAMPTHRH3
SCHEMBL6563410 0.84 GAA (0.40) GAAALDH1A1HPGDNAMPTHSD11B1
SCHEMBL6561835 0.84 PTPN11 (0.35) GAAALDH1A1HPGDNAMPTNPC1
SCHEMBL6565309 0.81 PTPN11 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed