SCHEMBL6563507

SCHEMBL6563507

CCOC(=O)Cc1cc(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)c(C)cc1C(=O)N1CCCC1C

nearest known ligand 0.31

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 4/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
TSHR P16473 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.30
HSD11B1 P28845 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
NAMPT P43490 1/20 0.30
HTT P42858 1/20 0.30
NPC1 O15118 1/20 0.30
ACHE P22303 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563752 0.90 GAA (0.35) KCNK3MEN1KMT2ATSHRALDH1A1
SCHEMBL6561673 0.87 PRSS1 (0.35) MEN1KMT2ATSHRALDH1A1GAA
SCHEMBL6563605 0.85 GAA (0.37) MEN1KMT2AALDH1A1GAAHPGD
SCHEMBL6565417 0.83 PTPN11 (0.36) KCNK3ALDH1A1GAAHPGDHSD11B1
SCHEMBL6561843 0.82 GAA (0.31) MEN1KMT2ATSHRGAAHSD11B1
SCHEMBL6561835 0.80 PTPN11 (0.35) KCNK3MEN1KMT2AALDH1A1GAA
SCHEMBL6563002 0.79 HRH3 (0.42) ALDH1A1GAAHPGDHSD11B1HRH3
SCHEMBL6563591 0.79 LRRK2 (0.39) MEN1KMT2AALDH1A1GAAHPGD
SCHEMBL6565367 0.79 TSHR (0.31) MEN1KMT2ATSHR
SCHEMBL6563779 0.79 KCNK3 (0.38) KCNK3MEN1KMT2AGAAHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed