SCHEMBL6565403

SCHEMBL6565403

O=C(c1ccc(C#CCNc2ccccc2)cc1)c1cccs1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.54
HPGD P15428 5/20 0.50
RAB9A P51151 5/20 0.50
NPC1 O15118 4/20 0.50
TSHR P16473 1/20 0.50
CYP2C9 P11712 3/20 0.47
LMNA P02545 3/20 0.47
ALDH1A1 P00352 3/20 0.47
PTGS1 P23219 2/20 0.47
PTGS2 P35354 2/20 0.47
KDM4E B2RXH2 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
HTT P42858 2/20 0.47
EGLN1 Q9GZT9 1/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALOX15 P16050 1/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
PGR P06401 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561875 0.89 HPGD (0.47) HPGDSHPGDRAB9ANPC1TSHR
SCHEMBL7670097 0.87 HPGD (0.45) HPGDSHPGDRAB9ANPC1TSHR
SCHEMBL6563325 0.81 KMT2A (0.50) HPGDRAB9ACYP2C9LMNAALDH1A1
SCHEMBL29712728 0.78 SMN1; SMN2 (0.50) HPGDRAB9ANPC1LMNAALDH1A1
SCHEMBL28782860 0.76 CA1 (0.56) HPGDRAB9ANPC1TSHRCYP2C9
SCHEMBL6563532 0.75 ALDH1A1 (0.44) HPGDRAB9ANPC1LMNAALDH1A1
SCHEMBL6564996 0.75 KMT2A (0.54) HPGDRAB9ANPC1LMNAALDH1A1
SCHEMBL6563589 0.74 GALR3 (0.50) RAB9ACYP2C9LMNAALDH1A1EGLN1
SCHEMBL6565427 0.74 VNN1 (0.46) RAB9ANPC1EGLN1MEN1KMT2A
SCHEMBL11133426 0.74 PTPN11 (0.47) RAB9ANPC1TSHRCYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed