SCHEMBL6561875

SCHEMBL6561875

N#Cc1ccc(NCC#Cc2ccc(C(=O)c3cccs3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
TSHR P16473 1/20 0.47
PGR P06401 1/20 0.46
HTT P42858 2/20 0.44
HPGDS O60760 1/20 0.43
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 4/20 0.41
LMNA P02545 3/20 0.41
PTGS2 P35354 3/20 0.41
CYP2C9 P11712 2/20 0.41
PTGS1 P23219 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MAPT P10636 3/20 0.41
MELK Q14680 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565403 0.89 HPGDS (0.54) HPGDNPC1RAB9ATSHRPGR
SCHEMBL7670097 0.86 HPGD (0.45) HPGDNPC1RAB9ATSHRHTT
SCHEMBL6563532 0.83 ALDH1A1 (0.44) HPGDNPC1RAB9AHTTMEN1
SCHEMBL12714962 0.82 HPGDS (0.62) HPGDNPC1RAB9ATSHRPGR
SCHEMBL6565480 0.80 GSK3B (0.47) ALDH1A1LMNASMN1; SMN2
SCHEMBL6563651 0.78 MAPK13 (0.45) NPC1RAB9AHTTMEN1KMT2A
SCHEMBL6565408 0.76 CNR1 (0.41) HPGDNPC1RAB9AHTTMEN1
SCHEMBL6565461 0.76 VNN1 (0.48) TSHRPGRHTTMEN1KMT2A
SCHEMBL6565441 0.76 KMT2A (0.46) HPGDNPC1RAB9AHTTMEN1
SCHEMBL6563777 0.75 GSK3B (0.45) MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed