SCHEMBL6565461

SCHEMBL6565461

N#Cc1ccc(NCC#Cc2ccc(C(=O)c3cccc(Cl)c3)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 6/20 0.48
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
MAOB P27338 1/20 0.41
SIRT2 Q8IXJ6 3/20 0.41
PGR P06401 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
GRM5 P41594 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565427 0.90 VNN1 (0.46) VNN1MEN1KMT2APGREGLN1
SCHEMBL6563532 0.87 ALDH1A1 (0.44) VNN1MEN1KMT2AEGLN1LMNA
SCHEMBL7675043 0.87 F7 (0.42) VNN1PGREGLN1GRM5
SCHEMBL6565480 0.82 GSK3B (0.47) VNN1TDP1LMNA
SCHEMBL6564223 0.79 VNN1 (0.41) VNN1MEN1KMT2AEGLN1LMNA
SCHEMBL6563213 0.77 KMT2A (0.39) VNN1MEN1KMT2ACYP11B1CYP11B2
SCHEMBL6563651 0.77 MAPK13 (0.45) MEN1KMT2ACYP11B1CYP11B2EGLN1
SCHEMBL6561875 0.76 HPGD (0.47) MEN1CYP2C9CYP2C19KMT2APGR
SCHEMBL6565408 0.75 CNR1 (0.41) VNN1MEN1KMT2ALMNAMAPT
SCHEMBL6565441 0.75 KMT2A (0.46) VNN1MEN1KMT2AEGLN1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed