SCHEMBL78404

SCHEMBL78404

CCC1=C(c2ccc(O)cc2)CC(CO[Si](C)(C)C(C)(C)C)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
HTR2C P28335 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
PREP P48147 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
AGTR2 P50052 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78635 0.90 PDK1 (0.35) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL65685 0.88 CHRM5 (0.40) PDK1PDK2PDK3PDK4CHRM2
SCHEMBL78854 0.85 PPARG (0.40) MEN1KMT2A
SCHEMBL78724 0.85 KDM4E (0.34) CHRM5CHRM1
SCHEMBL8701756 0.82 PSEN1 (0.41) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL8701755 0.82 PSEN1 (0.41) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL78407 0.81 PDK1 (0.37) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL7576828 0.81 PDK1 (0.40) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL65202 0.79 MGLL (0.36) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL91250 0.79 PARP1 (0.34) PDK1PDK2PDK3PDK4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed