SCHEMBL65202

SCHEMBL65202

CC(C)(C)[Si](C)(C)OCC1CC(c2cccc(-c3ccccc3)c2)=C(C(=O)O)CN1C(=O)OCc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.36
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
PPARA Q07869 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
POLB P06746 1/20 0.33
HTR2C P28335 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65231 0.92 CHRM5 (0.39) MGLLPDK1PDK2PDK3PDK4
SCHEMBL78635 0.90 PDK1 (0.35) MGLLPDK1PDK2PDK3PDK4
SCHEMBL78366 0.87 PDK1 (0.33) PDK1PDK2PDK3PDK4NPSR1
SCHEMBL91260 0.85 PPARA (0.35) MGLLPDK1PDK2PDK3PDK4
SCHEMBL65367 0.82 REN (0.38)
SCHEMBL64503 0.82 PPARA (0.33) PPARACHRM5CHRM1KDM4E
SCHEMBL64061 0.82 CHRM2 (0.38) PDK1PDK2PDK3PDK4CHRM2
SCHEMBL65685 0.81 CHRM5 (0.40) PDK1PDK2PDK3PDK4CHRM2
SCHEMBL65792 0.81 PPARA (0.39) PPARACHRM5CHRM1KDM4EALDH1A1
SCHEMBL8701755 0.80 PSEN1 (0.41) PDK1PDK2PDK3PDK4NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed