SCHEMBL6572500

SCHEMBL6572500

COCCN(CCOC)c1ccc(N)c(-c2cccc(Cl)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.40
CRHR1 P34998 3/20 0.38
PGR P06401 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36
TDO2 P48775 1/20 0.36
SLC6A9 P48067 1/20 0.35
BACE1 P56817 1/20 0.35
DHFR P00374 1/20 0.35
TP53 P04637 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
FYN P06241 1/20 0.34
RORC P51449 1/20 0.34
RORB Q92753 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34
STK4 Q13043 1/20 0.34
STK3 Q13188 1/20 0.34
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572811 0.88 CRHR1 (0.37) MAPTCRHR1MEN1KMT2A
SCHEMBL6571371 0.87 MAOA (0.34) FYN
SCHEMBL6572821 0.86 ALDH1A1 (0.37) MAPTCRHR1KMT2AFYNADORA2A
SCHEMBL6574166 0.86 MAP4K4 (0.42) MEN1KMT2AFYNTAAR1
SCHEMBL6574728 0.85 KMT2A (0.41) CRHR1TP53MEN1KMT2A
SCHEMBL6571441 0.85 CYP3A4 (0.38) FYNSTK3ADORA1
SCHEMBL6570969 0.85 ADK (0.36) MAPTCRHR1MEN1KMT2AADORA2A
SCHEMBL6572429 0.85 TDO2 (0.42) MAPTTDO2KMT2AADORA2AADORA1
SCHEMBL6571313 0.84 FYN (0.38) CRHR1MEN1KMT2AFYN
SCHEMBL6571876 0.83 CYP3A4 (0.40) CRHR1DHFRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed