SCHEMBL6584980

SCHEMBL6584980

O=C1Cc2c(cccc2OCCCN2CCN(Cc3ccc4ccccc4n3)CC2)N1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.45
DRD3 P35462 3/20 0.45
DRD4 P21917 2/20 0.45
HTR1A P08908 2/20 0.44
HTR7 P34969 1/20 0.44
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
ADRA1A P35348 1/20 0.42
FAAH O00519 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6586848 0.91 HTR1A (0.42) DRD2HTR1AHTR7MEN1MAPT
SCHEMBL6584734 0.89 HTR1A (0.41) DRD2HTR1AHTR7MEN1MAPT
SCHEMBL6583227 0.84 HTR1A (0.44) DRD2DRD3HTR1AHTR7MEN1
SCHEMBL6586928 0.82 MAOA (0.45) DRD2DRD3DRD4HTR1AHTR7
SCHEMBL8310206 0.81 HTR1A (0.42) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6585521 0.80 HTR1A (0.42) DRD2HTR1AHTR7MEN1MAPT
SCHEMBL8310251 0.80 DRD2 (0.46) DRD2DRD3DRD4HTR1AHTR7
SCHEMBL6581869 0.79 HTR1A (0.43) DRD2DRD3HTR1AHTR7MEN1
SCHEMBL6584872 0.79 DRD2 (0.48) DRD2HTR1A
SCHEMBL6582486 0.78 DRD2 (0.41) DRD2HTR1AHTR7MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed