SCHEMBL6586848

SCHEMBL6586848

O=C1CCCc2c(cccc2OCCCN2CCN(Cc3ccc4ccccc4n3)CC2)N1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.42
HTR7 P34969 1/20 0.42
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD2 P14416 2/20 0.40
HTR2A P28223 2/20 0.40
FAAH O00519 2/20 0.39
HCRTR1 O43613 3/20 0.39
HCRTR2 O43614 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584734 0.98 HTR1A (0.41) HTR1AHTR7MAOAMAOBMEN1
SCHEMBL6584980 0.91 DRD2 (0.45) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL6586928 0.83 MAOA (0.45) HTR1AHTR7MAOAMAOBMEN1
SCHEMBL6584542 0.82 DRD2 (0.56) HTR1AHTR7MAOAMAOBDRD2
SCHEMBL6585521 0.82 HTR1A (0.42) HTR1AHTR7MAOAMAOBMEN1
SCHEMBL8310251 0.82 DRD2 (0.46) HTR1AHTR7MAOAMAOBMEN1
SCHEMBL6582486 0.82 DRD2 (0.41) HTR1AHTR7MAOAMAOBMEN1
SCHEMBL6583227 0.81 HTR1A (0.44) HTR1AHTR7MEN1MAPTKMT2A
SCHEMBL8308852 0.81 DRD2 (0.54) HTR1AHTR7MAOAMAOBDRD2
SCHEMBL8310206 0.80 HTR1A (0.42) HTR1AHTR7MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed