SCHEMBL6586359

SCHEMBL6586359

N[C@@H](Cc1ccccc1)CN1CCN(c2nsnc2Cl)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.58
SLC6A4 P31645 4/20 0.43
SLC6A3 Q01959 4/20 0.43
AKT1 P31749 1/20 0.38
EPHX1 P07099 1/20 0.38
ALDH1A1 P00352 2/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
SLC6A2 P23975 2/20 0.37
SMO Q99835 1/20 0.37
HTR3E A5X5Y0 2/20 0.36
HTR3B O95264 2/20 0.36
HTR2C P28335 2/20 0.36
HTR3A P46098 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL6592709 0.92 HTR1A (0.58) HTR1ASLC6A4SLC6A3AKT1SLC6A2
SCHEMBL6589366 0.83 HTR1A (0.61) HTR1AAKT1DRD4DRD3
SCHEMBL6586745 0.76 HTR1A (0.48) HTR1AALDH1A1ALOX15TSHRMAPK1
SCHEMBL6586750 0.76 SIGMAR1 (0.58) ALDH1A1KDM4E
SCHEMBL13405022 0.76 DRD4 (0.57) HTR1ASLC6A4SLC6A3EPHX1ALDH1A1
SCHEMBL31232789 0.76 DRD4 (0.57) HTR1ASLC6A4SLC6A3EPHX1ALDH1A1
SCHEMBL6706541 0.75 SIGMAR1 (0.62) SLC6A4SLC6A3EPHX1ALDH1A1KDM4E
SCHEMBL6590854 0.74 HTR1A (1.00) HTR1AMAPK1DRD4DRD3
SCHEMBL27489107 0.74 HTR1A (1.00) HTR1AMAPK1DRD4DRD3
SCHEMBL4555805 0.72 MAPT (0.48) HTR1AALDH1A1ALOX15TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161424-B1 NEW DIAZOLE DERIVATIVES AS SEROTONERGIC AGENTS WYETH CORP (US) 2004-06-02 EP claimed
US-6239134-B1 TREATING CENTRAL NERVOUS SYSTEM DISORDERS USING THESE COMPOUNDS. NOVEL DIAZOLEPIPERAZINE, DIAZOLEPIPERIDINE, AND DIAZOLEDIHYDROPIPERIDINE DERIVATIVES, AMERICAN HOME PRODUCTS CORP. 2001-05-29 US claimed