SCHEMBL658682

SCHEMBL658682

NC(=O)Cc1ccc2c(c1)OCCCO2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
RAB9A P51151 5/20 0.52
HPGD P15428 3/20 0.52
USP2 O75604 1/20 0.52
LMNA P02545 1/20 0.52
GAA P10253 1/20 0.52
ALOX15 P16050 1/20 0.52
HTT P42858 1/20 0.52
HSD17B10 Q99714 1/20 0.52
CYP3A4 P08684 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
MAPK8 P45983 2/20 0.50
NPSR1 Q6W5P4 1/20 0.49
TSHR P16473 1/20 0.49
NPC1 O15118 5/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CASP3 P42574 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3525050 0.93 ALDH1A1 (0.59) ALDH1A1RAB9AHPGDUSP2LMNA
SCHEMBL1395778 0.86 CYP3A4 (0.68) ALDH1A1RAB9AHPGDLMNACYP3A4
SCHEMBL31409465 0.85 ALDH1A1 (0.57) ALDH1A1RAB9AHPGDUSP2LMNA
Hydrochloric Acid SCHEMBL6296149 0.85 CYP3A4 (0.66) ALDH1A1RAB9AHPGDLMNACYP3A4
SCHEMBL30232548 0.83 CYP3A4 (0.51) ALDH1A1RAB9AHPGDUSP2LMNA
SCHEMBL5792636 0.83 CTNNB1 (0.50) ALDH1A1RAB9AHPGDUSP2LMNA
SCHEMBL2777357 0.80 RAB9A (0.52) RAB9ANPC1SMN1; SMN2CASP3CA2
SCHEMBL31409466 0.80 SMN1; SMN2 (0.51) ALDH1A1RAB9AHPGDUSP2LMNA
SCHEMBL1468159 0.79 ALDH1A1 (0.62) ALDH1A1RAB9AHPGDUSP2LMNA
SCHEMBL286952 0.77 ALDH1A1 (0.60) ALDH1A1RAB9AHPGDUSP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10703754-B2 Compounds and compositions for treating chemical warfare agent-induced injuries ELI LILLY AND COMPANY (US) 2020-07-07 US disclosed
US-20190194202-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES ELI LILLY AND COMPANY 2019-06-27 US disclosed
US-20180265511-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES ELI LILLY AND COMPANY 2018-09-20 US disclosed
US-20180133170-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS ELI LILLY AND COMPANY 2018-05-17 US disclosed
US-20130059869-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS HYDRA BIOSCIENCES, INC. 2013-03-07 US disclosed
US-20120046305-A1 METHODS AND COMPOSITIONS FOR TREATING RESPIRATORY DISORDERS ELI LILLY AND COMPANY 2012-02-23 US disclosed
US-20090143377-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS ELI LILLY AND COMPANY 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10703754-B2 Compounds and compositions for treating chemical warfare agent-induced injuries ELANE, CASP3, MMP8 ALDH1A1 1104/4885RAB9A 1580/4885HPGD 1082/4885
US-20180133170-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 ALDH1A1 968/4885RAB9A 2306/4885HPGD 1228/4885
US-20180265511-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES ELANE, CASP3, MMP8 ALDH1A1 1104/4885RAB9A 1580/4885HPGD 1082/4885
US-20090143377-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 ALDH1A1 968/4885RAB9A 2306/4885HPGD 1228/4885
US-20120046305-A1 METHODS AND COMPOSITIONS FOR TREATING RESPIRATORY DISORDERS TRPA1, TRPV1, TRPV3 ALDH1A1 1173/4885RAB9A 2725/4885HPGD 584/4885
US-20190194202-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES ELANE, CASP3, MMP8 ALDH1A1 1104/4885RAB9A 1580/4885HPGD 1082/4885
US-20130059869-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 ALDH1A1 968/4885RAB9A 2306/4885HPGD 1228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.