SCHEMBL6586959

SCHEMBL6586959

Cn1cc(-c2nc3c(OC(N)=O)cccc3[nH]2)c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
ALDH1A1 P00352 2/20 0.56
HPGD P15428 2/20 0.56
TSHR P16473 2/20 0.56
HSD17B10 Q99714 2/20 0.56
NPC1 O15118 1/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56
HTT P42858 1/20 0.56
RAB9A P51151 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
PARP1 P09874 4/20 0.47
GRK2 P25098 1/20 0.42
CDC7 O00311 1/20 0.42
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587773 0.88 PARP1 (0.46) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL6806945 0.84 PARP1 (0.60) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL6589817 0.83 PIM1 (0.41) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL6590569 0.81 L3MBTL1 (0.48) KDM4EPARP1
SCHEMBL6588173 0.79 PARP1 (0.49) ALDH1A1PARP1MEN1KMT2A
SCHEMBL6588299 0.76 PARP1 (0.47) ALDH1A1NPC1MAPTSMN1; SMN2PARP1
SCHEMBL6587182 0.76 MEN1 (0.52) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL6587303 0.75 EPHX2 (0.52) PARP1
SCHEMBL7479706 0.74 PARP1 (0.49) PARP1
SCHEMBL6587520 0.73 PARP1 (0.46) ALDH1A1NPC1LMNAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed